Compile Data Set for Download or QSAR
Found 248 from Glaxo Wellcome
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50038168(7-Chloro-4-hydroxy-3-(3-phenoxy-phenyl)-1H-quinoli...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471539(CHEMBL117627)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471520(CHEMBL117691)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471528(CHEMBL168394)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471526(GAVESTINEL SODIUM | Gavestinel)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471538(CHEMBL168754)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471521(CHEMBL355109)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471544(CHEMBL166552)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471522(CHEMBL433725)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471550(CHEMBL169566)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471549(CHEMBL262537)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471548(CHEMBL354980)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50005075((2R,4S)-5,7-Dichloro-4-(3-phenyl-ureido)-1,2,3,4-t...)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471537(CHEMBL168465)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471534(CHEMBL168470)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50038161(6,7-Dichloro-3-hydroxy-5-nitro-3,4-dihydro-1H-quin...)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471540(CHEMBL169013)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471541(CHEMBL354793)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471535(CHEMBL169368)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471547(CHEMBL168503)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471530(CHEMBL168828)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471551(CHEMBL352435)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471524(CHEMBL169227)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471532(CHEMBL169776)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471523(CHEMBL354484)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471536(CHEMBL353977)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471545(CHEMBL353272)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471525(CHEMBL352310)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471543(CHEMBL323628)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471533(CHEMBL354375)copy SMILEScopy InChI
Affinity DataKi:  126nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471531(CHEMBL169890)copy SMILEScopy InChI
Affinity DataKi:  158nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471542(CHEMBL355298)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471529(CHEMBL435473)copy SMILEScopy InChI
Affinity DataKi:  501nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471546(CHEMBL352828)copy SMILEScopy InChI
Affinity DataKi:  794nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Glaxo Wellcome S.p.A.

Curated by ChEMBL
LigandPNGBDBM50471527(CHEMBL168924)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of [3H]glycine to glycine binding site, associated with the N-methyl-D-aspartate glutamate receptor 1 in crude synaptic membranes prepared...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5JBVPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50036918(2-[4-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-bu...)copy SMILEScopy InChI
Affinity DataIC50: 0.190nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding at serotonin 5-hydroxytryptamine 1A receptor from rat hippocampus tissue.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ60MNPubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Glaxo Wellcome

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMAssay Description:Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor stably expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3SZ1PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50051280(CHEMBL544436 | N-[4-(4-Benzo[d]isothiazol-3-yl-pip...)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:In vitro inhibitory activity against [3H]raclopride binding to dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ912QPubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Glaxo Wellcome

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 0.630nMAssay Description:Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3SZ1PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50051285(CHEMBL542554 | {4-[4-(4-Benzo[d]isothiazol-3-yl-pi...)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibitory activity against [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ912QPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50048817(2-[6-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-he...)copy SMILEScopy InChI
Affinity DataIC50: 0.760nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding at serotonin 5-hydroxytryptamine 1A receptor from rat hippocampus tissue.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ60MNPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50051286(CHEMBL544434 | N-[4-(4-Benzo[d]isothiazol-3-yl-pip...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity against [3H]raclopride binding to dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ912QPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50051277(2-Amino-N-[4-(4-benzo[d]isothiazol-3-yl-piperazin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:In vitro inhibitory activity against [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ912QPubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50054718(3-Amino-thiophene-2-carboxylic acid [4-(4-benzo[d]...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1R6TPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50051257(CHEMBL545607 | N-[4-(4-Benzo[d]isothiazol-3-yl-pip...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:In vitro inhibitory activity against [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ912QPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50051259(2-Amino-N-[4-(4-benzo[d]isothiazol-3-yl-piperazin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity against [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ912QPubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50054710(1,2,3,4-Tetrahydro-quinoline-8-carboxylic acid [4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1R6TPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50048818(2-[5-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-pe...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding at serotonin 5-hydroxytryptamine 1A receptor from rat hippocampus tissue.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ60MNPubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50054713(2-Amino-thiophene-3-carboxylic acid [4-(4-benzo[d]...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1R6TPubMed
TargetD(2) dopamine receptor(Mus musculus (Mouse))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50054716(1H-Indazole-3-carboxylic acid [4-(4-benzo[d]isothi...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of mouse Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1R6TPubMed
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